Detalhe da pesquisa
1.
Firefly luciferase inhibitor-conjugated peptide quenches bioluminescence: a versatile tool for real time monitoring cellular uptake of biomolecules.
Bioconjug Chem
; 25(1): 4-10, 2014 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-24341748
2.
Synthesis and biological evaluation of phenolic 4,5-dihydroisoxazoles and 3-hydroxy ketones as estrogen receptor alpha and beta agonists.
Bioorg Med Chem
; 18(10): 3437-47, 2010 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20430632
3.
Synthesis and evaluation of estrogen agonism of diaryl 4,5-dihydroisoxazoles, 3-hydroxyketones, 3-methoxyketones, and 1,3-diketones: a compound set forming a 4D molecular library.
J Med Chem
; 51(12): 3562-71, 2008 Jun 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-18517258
4.
Improved assays for xenosensor activation based on reverse transfection.
Toxicol In Vitro
; 29(7): 1759-65, 2015 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-26187274
5.
Synthesis and biological evaluation of second-generation tropanol-based androgen receptor modulators.
J Med Chem
; 58(3): 1569-74, 2015 Feb 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-25646649
6.
Preclinical pharmacology of FL442, a novel nonsteroidal androgen receptor modulator.
Mol Cell Endocrinol
; 387(1-2): 8-18, 2014 Apr 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-24565895
7.
Discovery of 5-benzyl-3-phenyl-4,5-dihydroisoxazoles and 5-benzyl-3-phenyl-1,4,2-dioxazoles as potent firefly luciferase inhibitors.
J Med Chem
; 56(3): 1064-73, 2013 Feb 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-23286196
8.
Design, synthesis, and biological evaluation of nonsteroidal cycloalkane[d]isoxazole-containing androgen receptor modulators.
J Med Chem
; 55(14): 6316-27, 2012 Jul 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-22746350
9.
Ligand specificity of constitutive androstane receptor as probed by induced-fit docking and mutagenesis.
J Med Chem
; 51(22): 7119-31, 2008 Nov 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-18973326