Detalhe da pesquisa
1.
Synthesis and structure activity relationship of imidazo[1,2-a]pyridine-8-carboxamides as a novel antimycobacterial lead series.
Bioorg Med Chem Lett
; 23(17): 4996-5001, 2013 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23867166
2.
Novel N-linked aminopiperidine-based gyrase inhibitors with improved hERG and in vivo efficacy against Mycobacterium tuberculosis.
J Med Chem
; 57(11): 4889-905, 2014 Jun 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-24809953
3.
Aminopyrazinamides: novel and specific GyrB inhibitors that kill replicating and nonreplicating Mycobacterium tuberculosis.
ACS Chem Biol
; 8(3): 519-23, 2013 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23268609
4.
Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B.
J Med Chem
; 56(21): 8834-48, 2013 Nov 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-24088190