Detalhe da pesquisa
1.
Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure-activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-ß-D-ribose 2'-oxidase.
Bioorg Med Chem
; 23(24): 7694-710, 2015 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-26643218
2.
Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis.
J Med Chem
; 60(4): 1379-1399, 2017 02 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-28075132
3.
Genetic and chemical validation identifies Mycobacterium tuberculosis topoisomerase I as an attractive anti-tubercular target.
Tuberculosis (Edinb)
; 95(5): 589-98, 2015 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-26073894
4.
Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate.
Nat Commun
; 6: 6715, 2015 Mar 31.
Artigo
em Inglês
| MEDLINE | ID: mdl-25823686
5.
Discovery of pyrazolopyridones as a novel class of noncovalent DprE1 inhibitor with potent anti-mycobacterial activity.
J Med Chem
; 57(11): 4761-71, 2014 Jun 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-24818517
6.
4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity.
J Med Chem
; 57(12): 5419-34, 2014 Jun 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-24871036
7.
Aminoazabenzimidazoles, a novel class of orally active antimalarial agents.
J Med Chem
; 57(13): 5702-13, 2014 Jul 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-24914738
8.
Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B.
J Med Chem
; 56(21): 8834-48, 2013 Nov 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-24088190