Detalhe da pesquisa
1.
Development of Endocyclic Control Elements for Peptide Macrocycles.
J Am Chem Soc
; 140(28): 8763-8770, 2018 07 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-29920073
2.
The effect of backbone flexibility on site-selective modification of macrocycles.
Org Biomol Chem
; 14(43): 10230-10237, 2016 Nov 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-27735955
3.
Synthesis of Aminoboronic Acid Derivatives from Amines and Amphoteric Boryl Carbonyl Compounds.
Angew Chem Int Ed Engl
; 55(41): 12659-63, 2016 10 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-27584917
4.
Solid-Phase Parallel Synthesis of Functionalised Medium-to-Large Cyclic Peptidomimetics through Three-Component Coupling Driven by Aziridine Aldehyde Dimers.
Chemistry
; 21(25): 9249-55, 2015 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-26014974
5.
Potent complement C3a receptor agonists derived from oxazole amino acids: Structure-activity relationships.
Bioorg Med Chem Lett
; 25(23): 5604-8, 2015 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26522948
6.
Site-specific integration of amino acid fragments into cyclic peptides.
J Am Chem Soc
; 136(10): 3728-31, 2014 Mar 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-24533886
7.
Stereocontrolled disruption of the Ugi reaction toward the production of chiral piperazinones: substrate scope and process development.
J Org Chem
; 79(21): 9948-57, 2014 Nov 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-25254948
8.
Conformational modulation of in vitro activity of cyclic RGD peptides via aziridine aldehyde-driven macrocyclization chemistry.
Bioconjug Chem
; 23(7): 1387-95, 2012 Jul 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-22709546
9.
Bending rigid molecular rods: formation of oligoproline macrocycles.
Chemistry
; 18(49): 15612-7, 2012 Dec 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-23124621
10.
Recent Developments in Therapeutic Peptides for the Glucagon-like Peptide 1 and 2 Receptors.
J Med Chem
; 63(3): 905-927, 2020 02 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-31577440
11.
Advances in therapeutic peptides targeting G protein-coupled receptors.
Nat Rev Drug Discov
; 19(6): 389-413, 2020 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-32494050
12.
Metal clips that induce unstructured pentapeptides to be alpha-helical in water.
J Am Chem Soc
; 131(12): 4505-12, 2009 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-19317508
13.
Exocyclic control of turn induction in macrocyclic peptide scaffolds.
Chemistry
; 19(52): 17668-72, 2013 Dec 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-24259185
14.
Oxadiazole grafts in peptide macrocycles.
Nat Chem
; 8(12): 1105-1111, 2016 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-27874866
15.
The reactivity and conformational control of cyclic tetrapeptides derived from aziridine-containing amino acids.
Chem Sci
; 7(11): 6662-6668, 2016 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28567256
16.
Passive Membrane Permeability of Macrocycles Can Be Controlled by Exocyclic Amide Bonds.
J Med Chem
; 59(11): 5368-76, 2016 06 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-27120576
17.
Rational Design of Calpain Inhibitors Based on Calpastatin Peptidomimetics.
J Med Chem
; 59(11): 5403-15, 2016 06 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-27148623
18.
Facile synthesis of borofragments and their evaluation in activity-based protein profiling.
Chem Commun (Camb)
; 51(17): 3608-11, 2015 Feb 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-25633248
19.
Mechanistic investigation of aziridine aldehyde-driven peptide macrocyclization: the imidoanhydride pathway.
Chem Sci
; 6(10): 5446-5455, 2015 Oct 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29861887
20.
Development of the direct Suzuki-Miyaura cross-coupling of primary B-alkyl MIDA-boronates and aryl bromides.
Org Lett
; 16(5): 1338-41, 2014 Mar 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-24527782