Detalhe da pesquisa
1.
gamma-Secretase: characterization and implication for Alzheimer disease therapy.
Neurobiol Aging
; 23(6): 1023-30, 2002.
Artigo
em Inglês
| MEDLINE | ID: mdl-12470798
2.
Metabolism-directed optimization of 3-aminopyrazinone acetamide thrombin inhibitors. Development of an orally bioavailable series containing P1 and P3 pyridines.
J Med Chem
; 46(4): 461-73, 2003 Feb 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-12570369
3.
P2 pyridine N-oxide thrombin inhibitors: a novel peptidomimetic scaffold.
Bioorg Med Chem Lett
; 15(11): 2771-5, 2005 Jun 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-15911253
4.
Pharmacokinetic optimization of 3-amino-6-chloropyrazinone acetamide thrombin inhibitors. Implementation of P3 pyridine N-oxides to deliver an orally bioavailable series containing P1 N-benzylamides.
Bioorg Med Chem Lett
; 13(7): 1353-7, 2003 Apr 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-12657281