Detalhe da pesquisa
1.
Design, synthesis and molecular docking study of novel triazole-quinazolinone hybrids as antimalarial and antitubercular agents.
Bioorg Med Chem Lett
; 108: 129800, 2024 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-38763480
2.
Design, synthesis and antitubercular assessment of 1, 2, 3-triazole incorporated thiazolylcarboxylate derivatives.
Bioorg Med Chem Lett
; 97: 129551, 2024 01 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-37979730
3.
A Green one-pot three component synthesis of thiazolidine-2,4-dione based bisspirooxindolo-pyrrolidines with [Bmim]BF4: their in vitro and in silico anti-TB studies.
Mol Divers
; 2024 May 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-38789853
4.
Design, synthesis, anti-mycobacterial activity, molecular docking and ADME analysis of spiroquinoxaline-1,2,4-oxadiazoles via [3 + 2] cycloaddition reaction under ultrasound irradiation.
Mol Divers
; 2024 Jan 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-38261121
5.
N-Substituted piperazine-coupled imidazo[2,1-b]thiazoles as inhibitors of Mycobacterium tuberculosis: Synthesis, evaluation, and docking studies.
Drug Dev Res
; 85(1): e22153, 2024 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-38349258
6.
New tetrahydropyrimidine-1,2,3-triazole clubbed compounds: Antitubercular activity and Thymidine Monophosphate Kinase (TMPKmt) inhibition.
Bioorg Chem
; 131: 106312, 2023 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-36528922
7.
Synthesis, biological evaluation and molecular docking study of some new 4-aminosalicylic acid derivatives as anti-inflammatory and antimycobacterial agents.
Bioorg Chem
; 132: 106344, 2023 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-36669356
8.
Design and synthesis of novel quinazolinyl-bisspirooxindoles as potent anti-tubercular agents: an ultrasound-promoted methodology.
Mol Divers
; 27(3): 1427-1436, 2023 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-35933454
9.
Aryl-n-hexanamide linked enaminones of usnic acid as promising antimicrobial agents.
Mol Divers
; 27(2): 811-836, 2023 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-35608808
10.
First-in-class pyrido[2,3-d]pyrimidine-2,4(1H,3H)-diones against leishmaniasis and tuberculosis: Rationale, in vitro, ex vivo studies and mechanistic insights.
Arch Pharm (Weinheim)
; 355(4): e2100440, 2022 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-35106845
11.
Stereoselective synthesis and discovery of novel spirooxindolopyrrolidine engrafted indandione heterocyclic hybrids as antimycobacterial agents.
Bioorg Chem
; 110: 104798, 2021 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-33735710
12.
Design, synthesis, and biological evaluation of benzo[d]imidazole-2-carboxamides as new anti-TB agents.
Bioorg Chem
; 107: 104538, 2021 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-33349456
13.
Indole-fused spirochromenes as potential anti-tubercular agents: design, synthesis and in vitro evaluation.
Mol Divers
; 25(4): 2137-2148, 2021 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-32474889
14.
Design and characterisation of piperazine-benzofuran integrated dinitrobenzenesulfonamide as Mycobacterium tuberculosis H37Rv strain inhibitors.
J Enzyme Inhib Med Chem
; 36(1): 1751-1759, 2021 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-34325595
15.
Synthesis and antimicrobial evaluation of new nitric oxide-donating fluoroquinolone/oxime hybrids.
Arch Pharm (Weinheim)
; 354(1): e2000180, 2021 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-32959443
16.
Antihypernociceptive effects of Petersianthus macrocarpus stem bark on neuropathic pain induced by chronic constriction injury in rats.
Inflammopharmacology
; 29(4): 1241-1253, 2021 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-34081248
17.
Design and synthesis of purine connected piperazine derivatives as novel inhibitors of Mycobacterium tuberculosis.
Bioorg Med Chem Lett
; 30(22): 127512, 2020 11 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32871269
18.
Design and synthesis of new indanol-1,2,3-triazole derivatives as potent antitubercular and antimicrobial agents.
Bioorg Med Chem Lett
; 30(22): 127579, 2020 11 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32987135
19.
Novel isoniazid embedded triazole derivatives: Synthesis, antitubercular and antimicrobial activity evaluation.
Bioorg Med Chem Lett
; 30(19): 127434, 2020 10 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-32717369
20.
Synthesis and efficacy of pyrvinium-inspired analogs against tuberculosis and malaria pathogens.
Bioorg Med Chem Lett
; 30(8): 127037, 2020 04 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32081449