Detalhe da pesquisa
1.
Fast acting allosteric phosphofructokinase inhibitors block trypanosome glycolysis and cure acute African trypanosomiasis in mice.
Nat Commun
; 12(1): 1052, 2021 02 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-33594070
2.
New quinoline NK3 receptor antagonists with CNS activity.
Bioorg Med Chem Lett
; 19(3): 837-40, 2009 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-19117759
3.
Bifunctional crosslinking ligands for transthyretin.
Open Biol
; 5(9): 150105, 2015 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-26400472
4.
Design and synthesis of trans-3-(2-(4-((3-(3-(5-methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine (SB-414796): a potent and selective dopamine D3 receptor antagonist.
J Med Chem
; 46(23): 4952-64, 2003 11 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-14584946
5.
Discovery of 1-(3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-2-imidazolidinone (GSK163090), a Potent, selective, and orally active 5-HT1A/B/D receptor antagonist.
J Med Chem
; 53(23): 8228-40, 2010 Dec 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-21053897
6.
Studies on a series of potent, orally bioavailable, 5-HT(1) receptor ligands.
Bioorg Med Chem Lett
; 17(18): 5214-7, 2007 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-17629698
7.
3,4-Dihydro-2H-benzoxazinones as dual-acting 5-HT1A receptor antagonists and serotonin reuptake inhibitors.
Bioorg Med Chem Lett
; 17(4): 1033-6, 2007 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-17129726
8.
Tetrahydropyrido[3,4-b]pyrazine scaffolds from pentafluoropyridine.
J Org Chem
; 70(18): 7208-16, 2005 Sep 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-16122239
9.
Polyfunctional tetrahydropyrido[2,3-b]pyrazine scaffolds from 4-phenylsulfonyl tetrafluoropyridine.
J Org Chem
; 70(23): 9377-81, 2005 Nov 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-16268611
10.
3,4-Dihydro-2H-benzoxazinones are 5-HT(1A) receptor antagonists with potent 5-HT reuptake inhibitory activity.
Bioorg Med Chem Lett
; 15(3): 737-41, 2005 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-15664848