Detalhe da pesquisa
1.
Triphenylphosphonium conjugation to a TRAP1 inhibitor, 2-amino-6-chloro-7,9-dihydro-8H-purin-8-one increases antiproliferative activity.
Bioorg Chem
; 126: 105856, 2022 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-35661618
2.
Mitoquinone Inactivates Mitochondrial Chaperone TRAP1 by Blocking the Client Binding Site.
J Am Chem Soc
; 143(47): 19684-19696, 2021 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-34758612
3.
Discovery of 2-((4-resorcinolyl)-5-aryl-1,2,3-triazol-1-yl)acetates as potent Hsp90 inhibitors with selectivity over TRAP1.
Bioorg Med Chem Lett
; 30(2): 126809, 2020 01 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31839539
4.
Correction to "Mitoquinone Inactivates Mitochondrial Chaperone TRAP1 by Blocking the Client Binding Site".
J Am Chem Soc
; 144(4): 2020, 2022 Feb 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-35044746
5.
Design and Synthesis of TRAP1 Selective Inhibitors: H-Bonding with Asn171 Residue in TRAP1 Increases Paralog Selectivity.
ACS Med Chem Lett
; 12(7): 1173-1180, 2021 Jul 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-34267888