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Structure activity relationships of fused bicyclic and urea derivatives of spirocyclic compounds as potent CCR1 antagonists.
Hossain, Nafizal; Mensonides-Harsema, Marguérite; Cooper, Martin E; Eriksson, Tomas; Ivanova, Svetlana; Bergström, Lena.
Afiliação
  • Hossain N; Department of Medicinal Chemistry, Respiratory, Inflammation and Autoimmunity Innovative Medicines, AstraZeneca R&D, Pepparedsleden 1, SE-431 83 Mölndal, Sweden. Electronic address: nafizal.hossain@astrazeneca.com.
  • Mensonides-Harsema M; Department of Medicinal Chemistry, AstraZeneca R&D Lund, Scheelevägen 1, SE-221 87 Lund, Sweden.
  • Cooper ME; Department of Medicinal Chemistry, Respiratory, Inflammation and Autoimmunity Innovative Medicines, AstraZeneca R&D, Pepparedsleden 1, SE-431 83 Mölndal, Sweden.
  • Eriksson T; Department of Medicinal Chemistry, AstraZeneca R&D Lund, Scheelevägen 1, SE-221 87 Lund, Sweden.
  • Ivanova S; Department of Medicinal Chemistry, AstraZeneca R&D Lund, Scheelevägen 1, SE-221 87 Lund, Sweden.
  • Bergström L; Department of Medicinal Chemistry, Respiratory, Inflammation and Autoimmunity Innovative Medicines, AstraZeneca R&D, Pepparedsleden 1, SE-431 83 Mölndal, Sweden.
Bioorg Med Chem Lett ; 24(1): 108-12, 2014 Jan 01.
Article em En | MEDLINE | ID: mdl-24332486

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Compostos de Espiro / Ureia / Compostos Bicíclicos com Pontes / Receptores CCR1 Limite: Animals Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Compostos de Espiro / Ureia / Compostos Bicíclicos com Pontes / Receptores CCR1 Limite: Animals Idioma: En Ano de publicação: 2014 Tipo de documento: Article