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Structure-activity relationships and colorimetric properties of specific probes for the putative cancer biomarker human arylamine N-acetyltransferase 1.
Egleton, James E; Thinnes, Cyrille C; Seden, Peter T; Laurieri, Nicola; Lee, Siu Po; Hadavizadeh, Kate S; Measures, Angelina R; Jones, Alan M; Thompson, Sam; Varney, Amy; Wynne, Graham M; Ryan, Ali; Sim, Edith; Russell, Angela J.
Afiliação
  • Egleton JE; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK.
  • Thinnes CC; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK.
  • Seden PT; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.
  • Laurieri N; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK.
  • Lee SP; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK.
  • Hadavizadeh KS; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK.
  • Measures AR; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.
  • Jones AM; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.
  • Thompson S; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.
  • Varney A; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK.
  • Wynne GM; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK.
  • Ryan A; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK; Faculty of Science, Engineering and Computing, University of Kingston, KT1 2EE, UK.
  • Sim E; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK; Faculty of Science, Engineering and Computing, University of Kingston, KT1 2EE, UK.
  • Russell AJ; Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford OX1 3TA, UK; Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, UK. Electronic address: angela.russell@chem.ox.ac.uk.
Bioorg Med Chem ; 22(11): 3030-54, 2014 Jun 01.
Article em En | MEDLINE | ID: mdl-24758871

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Arilamina N-Acetiltransferase / Biomarcadores Tumorais / Naftoquinonas / Inibidores Enzimáticos / Isoenzimas Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Arilamina N-Acetiltransferase / Biomarcadores Tumorais / Naftoquinonas / Inibidores Enzimáticos / Isoenzimas Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article