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Discovery and Hit-to-Lead Optimization of Non-ATP Competitive MK2 (MAPKAPK2) Inhibitors.
Huang, Xiaohua; Shipps, Gerald W; Cheng, Cliff C; Spacciapoli, Peter; Zhang, Xingmin; McCoy, Mark A; Wyss, Daniel F; Yang, Xianshu; Achab, Abdelghani; Soucy, Kyle; Montavon, Donna K; Murphy, Denise M; Whitehurst, Charles E.
Afiliação
  • Huang X; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Shipps GW; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Cheng CC; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Spacciapoli P; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Zhang X; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • McCoy MA; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Wyss DF; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Yang X; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Achab A; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Soucy K; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Montavon DK; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Murphy DM; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
  • Whitehurst CE; Merck Research Laboratories , 320 Bent Street, Cambridge, Massachusetts 02141, United States.
ACS Med Chem Lett ; 2(8): 632-7, 2011 Aug 11.
Article em En | MEDLINE | ID: mdl-24900358

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2011 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2011 Tipo de documento: Article