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Discovery of novel aromatase inhibitors using a homogeneous time-resolved fluorescence assay.
Ji, Jin-zi; Lao, Ke-jing; Hu, Jie; Pang, Tao; Jiang, Zhen-zhou; Yuan, Hao-liang; Miao, Jing-shan; Chen, Xin; Ning, Shan-shan; Xiang, Hua; Guo, Yu-meng; Yan, Ming; Zhang, Lu-yong.
Afiliação
  • Ji JZ; Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China.
  • Lao KJ; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Hu J; Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China.
  • Pang T; 1] Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China [2] Jiangsu Center for Pharmacodynamics Research and Evaluation, China Pharmaceutical University, Nanjing 210009, China.
  • Jiang ZZ; 1] Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China [2] Key Laboratory of Drug Quality Control and Pharmacovigilance (China Pharmaceutical University), Ministry of Education, Nanjing 210009, China.
  • Yuan HL; Laboratory of Molecular Design and Drug Discovery, School of Science, China Pharmaceutical University, Nanjing 210009, China.
  • Miao JS; Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China.
  • Chen X; Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China.
  • Ning SS; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Xiang H; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Guo YM; Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China.
  • Yan M; 1] Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China [2] Jiangsu Center for Pharmacodynamics Research and Evaluation, China Pharmaceutical University, Nanjing 210009, China.
  • Zhang LY; 1] Jiangsu Center for Drug Screening, China Pharmaceutical University, Nanjing 210009, China [2] State Key laboratory of Natural Medicines, China Pharmaceutical University, Nanjing 210009, China.
Acta Pharmacol Sin ; 35(8): 1082-92, 2014 Aug.
Article em En | MEDLINE | ID: mdl-25047514

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias da Mama / Ensaios de Seleção de Medicamentos Antitumorais / Inibidores da Aromatase / Bibliotecas de Moléculas Pequenas Limite: Female / Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias da Mama / Ensaios de Seleção de Medicamentos Antitumorais / Inibidores da Aromatase / Bibliotecas de Moléculas Pequenas Limite: Female / Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article