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Structural elucidation of the DFG-Asp in and DFG-Asp out states of TAM kinases and insight into the selectivity of their inhibitors.
Messoussi, Abdellah; Peyronnet, Lucile; Feneyrolles, Clémence; Chevé, Gwénaël; Bougrin, Khalid; Yasri, Aziz.
Afiliação
  • Messoussi A; OriBase Pharma, Parc Euromedecine, Cap Gamma, 1682, rue de la Valsière, 34189 Montpellier, France. khalid.bougrin@smct-ma.com.
  • Peyronnet L; OriBase Pharma, Parc Euromedecine, Cap Gamma, 1682, rue de la Valsière, 34189 Montpellier, France. lpeyronnet@oribase-pharma.com.
  • Feneyrolles C; OriBase Pharma, Parc Euromedecine, Cap Gamma, 1682, rue de la Valsière, 34189 Montpellier, France. cfeneyrolles@oribase-pharma.com.
  • Chevé G; OriBase Pharma, Parc Euromedecine, Cap Gamma, 1682, rue de la Valsière, 34189 Montpellier, France. gcheve@oribase-pharma.com.
  • Bougrin K; Laboratoire de Chimie des Plantes et de Synthèse Organique et Bioorganique, URAC23, Université Mohammed V, Faculté des Sciences B.P., 1014 Rabat, Morocco. khalid.bougrin@smct-ma.com.
  • Yasri A; OriBase Pharma, Parc Euromedecine, Cap Gamma, 1682, rue de la Valsière, 34189 Montpellier, France. ayasri@oribase-pharma.com.
Molecules ; 19(10): 16223-39, 2014 Oct 10.
Article em En | MEDLINE | ID: mdl-25310149

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores Proteína Tirosina Quinases / Inibidores de Proteínas Quinases Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores Proteína Tirosina Quinases / Inibidores de Proteínas Quinases Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article