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Engineering a Constrained Peptidic Scaffold towards Potent and Selective Furin Inhibitors.
Fittler, Heiko; Depp, Alexander; Avrutina, Olga; Dahms, Sven O; Than, Manuel E; Empting, Martin; Kolmar, Harald.
Afiliação
  • Fittler H; Clemens-Schöpf-Institut für organische und Biochemie, Technische Universität Darmstadt, Alarich-Weiss Strasse 4, 64287, Darmstadt, Germany.
  • Depp A; Clemens-Schöpf-Institut für organische und Biochemie, Technische Universität Darmstadt, Alarich-Weiss Strasse 4, 64287, Darmstadt, Germany.
  • Avrutina O; Clemens-Schöpf-Institut für organische und Biochemie, Technische Universität Darmstadt, Alarich-Weiss Strasse 4, 64287, Darmstadt, Germany.
  • Dahms SO; Leibniz Institute for Age Research-Fritz Lipmann Institute (FLI), Beutenbergstrasse 11, 07745, Jena, Germany.
  • Than ME; Leibniz Institute for Age Research-Fritz Lipmann Institute (FLI), Beutenbergstrasse 11, 07745, Jena, Germany.
  • Empting M; Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS), Campus C2.3, 66123, Saarbrücken, Germany.
  • Kolmar H; Clemens-Schöpf-Institut für organische und Biochemie, Technische Universität Darmstadt, Alarich-Weiss Strasse 4, 64287, Darmstadt, Germany. kolmar@biochemie-tud.de.
Chembiochem ; 16(17): 2441-4, 2015 Nov.
Article em En | MEDLINE | ID: mdl-26426719

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptídeos / Furina Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptídeos / Furina Idioma: En Ano de publicação: 2015 Tipo de documento: Article