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Y-shaped bis-arylethenesulfonic acid esters: Potential potent and membrane permeable protein tyrosine phosphatase 1B inhibitors.
Yang, Fengzhi; Xie, Fangzhou; Zhang, Ying; Xia, Yu; Liu, Wenlu; Jiang, Faqin; Lam, Celine; Qiao, Yixue; Xie, Dongsheng; Li, Jianqi; Fu, Lei.
Afiliação
  • Yang F; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China; China State Institute of Pharmaceutical Industry, Novel Technology Center of Pharmaceutical Chemistry, Shanghai Institute of Pharmaceutical Industry, Shanghai 201203, PR China.
  • Xie F; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China.
  • Zhang Y; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China.
  • Xia Y; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China; Viva Biotech (Shanghai) Limited, Shanghai 201203, PR China.
  • Liu W; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China.
  • Jiang F; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China.
  • Lam C; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China.
  • Qiao Y; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China.
  • Xie D; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China. Electronic address: dshxie@sjtu.edu.cn.
  • Li J; China State Institute of Pharmaceutical Industry, Novel Technology Center of Pharmaceutical Chemistry, Shanghai Institute of Pharmaceutical Industry, Shanghai 201203, PR China. Electronic address: li.jianqi@sipi.com.cn.
  • Fu L; School of Pharmacy, Shanghai Jiao Tong University, Shanghai 200240, PR China. Electronic address: leifu@sjtu.edu.cn.
Bioorg Med Chem Lett ; 27(10): 2166-2170, 2017 05 15.
Article em En | MEDLINE | ID: mdl-28372909

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Ácidos Sulfônicos / Inibidores Enzimáticos / Ésteres / Proteína Tirosina Fosfatase não Receptora Tipo 1 Tipo de estudo: Prognostic_studies Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Ácidos Sulfônicos / Inibidores Enzimáticos / Ésteres / Proteína Tirosina Fosfatase não Receptora Tipo 1 Tipo de estudo: Prognostic_studies Idioma: En Ano de publicação: 2017 Tipo de documento: Article