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Inhibition of bromodomain-containing protein 9 for the prevention of epigenetically-defined drug resistance.
Crawford, Terry D; Vartanian, Steffan; Côté, Alexandre; Bellon, Steve; Duplessis, Martin; Flynn, E Megan; Hewitt, Michael; Huang, Hon-Ren; Kiefer, James R; Murray, Jeremy; Nasveschuk, Christopher G; Pardo, Eneida; Romero, F Anthony; Sandy, Peter; Tang, Yong; Taylor, Alexander M; Tsui, Vickie; Wang, Jian; Wang, Shumei; Zawadzke, Laura; Albrecht, Brian K; Magnuson, Steven R; Cochran, Andrea G; Stokoe, David.
Afiliação
  • Crawford TD; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States. Electronic address: terrydc@gene.com.
  • Vartanian S; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Côté A; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Bellon S; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Duplessis M; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Flynn EM; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Hewitt M; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Huang HR; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Kiefer JR; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Murray J; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Nasveschuk CG; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Pardo E; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Romero FA; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Sandy P; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Tang Y; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Taylor AM; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Tsui V; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Wang J; Wuxi Apptec Co., Ltd., 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, PR China.
  • Wang S; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Zawadzke L; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Albrecht BK; Constellation Pharmaceuticals, 215 First Street, Suite 200, Cambridge, MA 02142, United States.
  • Magnuson SR; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Cochran AG; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States.
  • Stokoe D; Genentech Inc., 1 DNA Way, South San Francisco, CA 94080, United States. Electronic address: dhstokoe@calicolabs.com.
Bioorg Med Chem Lett ; 27(15): 3534-3541, 2017 08 01.
Article em En | MEDLINE | ID: mdl-28606761

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Resistência a Medicamentos / Epigênese Genética / Bibliotecas de Moléculas Pequenas Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Resistência a Medicamentos / Epigênese Genética / Bibliotecas de Moléculas Pequenas Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article