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Synthesis, antitumour and antioxidant activities of novel α,ß-unsaturated ketones and related heterocyclic analogues: EGFR inhibition and molecular modelling study.
El-Husseiny, Walaa M; El-Sayed, Magda A-A; Abdel-Aziz, Naglaa I; El-Azab, Adel S; Ahmed, Esam R; Abdel-Aziz, Alaa A-M.
Afiliação
  • El-Husseiny WM; a Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy , Mansoura University , Mansoura , Egypt.
  • El-Sayed MA; a Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy , Mansoura University , Mansoura , Egypt.
  • Abdel-Aziz NI; b Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Horus University , New Damietta , Egypt.
  • El-Azab AS; c Department of Medicinal Chemistry, Faculty of Pharmacy , Mansoura University , Mansoura , Egypt.
  • Ahmed ER; d Department of Pharmaceutical Chemistry, College of Pharmacy , King Saud University , Riyadh , Saudi Arabia.
  • Abdel-Aziz AA; e Department of Organic Chemistry, Faculty of Pharmacy , Al-Azhar University , Cairo , Egypt.
J Enzyme Inhib Med Chem ; 33(1): 507-518, 2018 Dec.
Article em En | MEDLINE | ID: mdl-29455554

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Proteínas Quinases / Receptores ErbB / Compostos Heterocíclicos / Cetonas / Antineoplásicos / Antioxidantes Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Proteínas Quinases / Receptores ErbB / Compostos Heterocíclicos / Cetonas / Antineoplásicos / Antioxidantes Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2018 Tipo de documento: Article