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The effect of elevated α1-acid glycoprotein on the pharmacokinetics of TAK-272 (SCO-272), an orally active renin inhibitor, in rats.
Ebihara, Takuya; Shimizu, Hisao; Yamamoto, Masami; Higuchi, Tomoaki; Jinno, Fumihiro; Tagawa, Yoshihiko.
Afiliação
  • Ebihara T; a Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division , Takeda Pharmaceutical Company Limited , Kanagawa , Japan.
  • Shimizu H; a Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division , Takeda Pharmaceutical Company Limited , Kanagawa , Japan.
  • Yamamoto M; a Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division , Takeda Pharmaceutical Company Limited , Kanagawa , Japan.
  • Higuchi T; a Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division , Takeda Pharmaceutical Company Limited , Kanagawa , Japan.
  • Jinno F; a Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division , Takeda Pharmaceutical Company Limited , Kanagawa , Japan.
  • Tagawa Y; a Drug Metabolism and Pharmacokinetics Research Laboratories, Pharmaceutical Research Division , Takeda Pharmaceutical Company Limited , Kanagawa , Japan.
Xenobiotica ; 49(5): 584-590, 2019 May.
Article em En | MEDLINE | ID: mdl-29790816

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piperidinas / Benzimidazóis / Orosomucoide / Morfolinas / Renina Limite: Animals Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piperidinas / Benzimidazóis / Orosomucoide / Morfolinas / Renina Limite: Animals Idioma: En Ano de publicação: 2019 Tipo de documento: Article