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Design, Synthesis, and Characterization of a Fluorescence Polarization Pan-BET Bromodomain Probe.
Paulson, Carolyn N; Guan, Xianghong; Ayoub, Alex M; Chan, Alice; Karim, Rezaul M; Pomerantz, William C K; Schönbrunn, Ernst; Georg, Gunda I; Hawkinson, Jon E.
Afiliação
  • Paulson CN; Department of Medicinal Chemistry and Institute for Therapeutics Discovery & Development, College of Pharmacy, University of Minnesota, 717 Delaware Street SE, Minneapolis, Minnesota 55414, United States.
  • Guan X; Department of Medicinal Chemistry and Institute for Therapeutics Discovery & Development, College of Pharmacy, University of Minnesota, 717 Delaware Street SE, Minneapolis, Minnesota 55414, United States.
  • Ayoub AM; Department of Chemistry, University of Minnesota, 207 Pleasant Street, SE, Minneapolis, Minnesota 55455, United States.
  • Chan A; H. Lee Moffitt Cancer Center & Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States.
  • Karim RM; Department of Molecular Medicine, University of South Florida, Tampa, Florida 33612, United States.
  • Pomerantz WCK; H. Lee Moffitt Cancer Center & Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States.
  • Schönbrunn E; Department of Molecular Medicine, University of South Florida, Tampa, Florida 33612, United States.
  • Georg GI; Department of Chemistry, University of Minnesota, 207 Pleasant Street, SE, Minneapolis, Minnesota 55455, United States.
  • Hawkinson JE; H. Lee Moffitt Cancer Center & Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States.
ACS Med Chem Lett ; 9(12): 1223-1229, 2018 Dec 13.
Article em En | MEDLINE | ID: mdl-30613330

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2018 Tipo de documento: Article