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Structure-based identification of novel CK2 inhibitors with a linear 2-propenone scaffold as anti-cancer agents.
Qi, Xiaoqian; Zhang, Na; Zhao, Lijiao; Hu, Liming; Cortopassi, Wilian A; Jacobson, Matthew P; Li, Xitao; Zhong, Rugang.
Afiliação
  • Qi X; Beijing Key Laboratory of Environmental & Viral Oncology, College of Life Science and Bioengineering, Beijing University of Technology, Beijing, 100124, China.
  • Zhang N; Beijing Key Laboratory of Environmental & Viral Oncology, College of Life Science and Bioengineering, Beijing University of Technology, Beijing, 100124, China. Electronic address: nanatonglei@bjut.edu.cn.
  • Zhao L; Beijing Key Laboratory of Environmental & Viral Oncology, College of Life Science and Bioengineering, Beijing University of Technology, Beijing, 100124, China.
  • Hu L; Beijing Key Laboratory of Environmental & Viral Oncology, College of Life Science and Bioengineering, Beijing University of Technology, Beijing, 100124, China.
  • Cortopassi WA; Department of Pharmaceutical Chemistry, University of California, San Francisco, CA, 94143, United States.
  • Jacobson MP; Department of Pharmaceutical Chemistry, University of California, San Francisco, CA, 94143, United States.
  • Li X; Shenzhen Grubbs Institute, Southern University of Science and Technology, Shenzhen, 518055, China.
  • Zhong R; Beijing Key Laboratory of Environmental & Viral Oncology, College of Life Science and Bioengineering, Beijing University of Technology, Beijing, 100124, China.
Biochem Biophys Res Commun ; 512(2): 208-212, 2019 04 30.
Article em En | MEDLINE | ID: mdl-30878184

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Caseína Quinase II / Inibidores de Proteínas Quinases / Antineoplásicos Tipo de estudo: Diagnostic_studies / Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Caseína Quinase II / Inibidores de Proteínas Quinases / Antineoplásicos Tipo de estudo: Diagnostic_studies / Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article