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Discovery of aromatic amides with triazole-core as potent reversal agents against P-glycoprotein-mediated multidrug resistance.
Qiu, Qianqian; Zhu, Jilan; Chen, Qiutong; Jiang, Ziqian; Xu, Jiting; Jiang, Xueting; Huang, Wenlong; Liu, Zhongquan; Ye, Jing; Xu, Xiaojuan.
Afiliação
  • Qiu Q; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China.
  • Zhu J; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China.
  • Chen Q; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China.
  • Jiang Z; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China.
  • Xu J; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China.
  • Jiang X; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China.
  • Huang W; Center of Drug Discovery, State Key Laboratory of Natural Medicines, China Pharmaceutical University, Nanjing, PR China; Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, China Pharmaceutical University, Nanjing, PR China.
  • Liu Z; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China. Electronic address: zhq6312@aliyun.com.
  • Ye J; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China. Electronic address: yej2017@163.com.
  • Xu X; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China. Electronic address: xuxj@yctu.edu.cn.
Bioorg Chem ; 90: 103083, 2019 09.
Article em En | MEDLINE | ID: mdl-31255991

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Triazóis / Benzamidas / Doxorrubicina / Membro 1 da Subfamília B de Cassetes de Ligação de ATP / Citocromo P-450 CYP3A / Amidas / Neoplasias / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Triazóis / Benzamidas / Doxorrubicina / Membro 1 da Subfamília B de Cassetes de Ligação de ATP / Citocromo P-450 CYP3A / Amidas / Neoplasias / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article