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Potently inhibiting cancer cell migration with novel 3H-pyrazolo[4,3-f]quinoline boronic acid ROCK inhibitors.
Dayal, Neetu; Mikek, Clinton G; Hernandez, Delmis; Naclerio, George A; Yin Chu, Elizabeth Fei; Carter-Cooper, Brandon A; Lapidus, Rena G; Sintim, Herman O.
Afiliação
  • Dayal N; Department of Chemistry, Purdue University, 560 Oval Drive, West Lafayette, IN, 47907, USA.
  • Mikek CG; Department of Chemistry, Purdue University, 560 Oval Drive, West Lafayette, IN, 47907, USA.
  • Hernandez D; Department of Chemistry, Purdue University, 560 Oval Drive, West Lafayette, IN, 47907, USA.
  • Naclerio GA; Department of Chemistry, Purdue University, 560 Oval Drive, West Lafayette, IN, 47907, USA.
  • Yin Chu EF; Department of Chemistry, Purdue University, 560 Oval Drive, West Lafayette, IN, 47907, USA.
  • Carter-Cooper BA; Translational Core Laboratory, University of Maryland Greenebaum Cancer Center, 655 W Baltimore Street, Baltimore, MD, 21201, USA.
  • Lapidus RG; Translational Core Laboratory, University of Maryland Greenebaum Cancer Center, 655 W Baltimore Street, Baltimore, MD, 21201, USA.
  • Sintim HO; Department of Chemistry, Purdue University, 560 Oval Drive, West Lafayette, IN, 47907, USA; Institute for Drug Discovery, Purdue University, 720 Clinic Drive, West Lafayette, IN, 47907, USA; Purdue Institute of Inflammation and Infectious Diseases, Purdue University, West Lafayette, IN, 47907, USA.
Eur J Med Chem ; 180: 449-456, 2019 Oct 15.
Article em En | MEDLINE | ID: mdl-31330446

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Ácidos Borônicos / Movimento Celular / Inibidores de Proteínas Quinases / Quinases Associadas a rho / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Ácidos Borônicos / Movimento Celular / Inibidores de Proteínas Quinases / Quinases Associadas a rho / Antineoplásicos Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article