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Discovery of tissue selective liver X receptor agonists for the treatment of atherosclerosis without causing hepatic lipogenesis.
Li, Chanjuan; Chen, Hao; Chen, Xinying; Li, Yanwen; Hua, Pei; Wei, Junkang; Song, Ching; Gu, Qiong; Zhou, Huihao; Zhang, Jingxia; Xu, Jun.
Afiliação
  • Li C; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Chen H; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Chen X; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Li Y; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Hua P; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Wei J; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Song C; School of Chemistry and Biological Engineering, University of Science and Technology Beijing, Beijing, 100083, China.
  • Gu Q; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Zhou H; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China.
  • Zhang J; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China. Electronic address: zhjingx@mail.sysu.edu.cn.
  • Xu J; School of Pharmaceutical Sciences, Sun Yat-Sen University, 132 East Circle Road at University City, Guangzhou, 510006, China. Electronic address: junxu@biochemomes.com.
Eur J Med Chem ; 182: 111647, 2019 Nov 15.
Article em En | MEDLINE | ID: mdl-31499362

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Esteróis / Aterosclerose / Descoberta de Drogas / Receptores X do Fígado Limite: Animals / Humans / Male Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Esteróis / Aterosclerose / Descoberta de Drogas / Receptores X do Fígado Limite: Animals / Humans / Male Idioma: En Ano de publicação: 2019 Tipo de documento: Article