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Antimigraine Drug Avitriptan Is a Ligand and Agonist of Human Aryl Hydrocarbon Receptor That Induces CYP1A1 in Hepatic and Intestinal Cells.
Vyhlídalová, Barbora; Krasulová, Kristýna; Pecinková, Petra; Poulíková, Karolína; Vrzal, Radim; Andrysík, Zdenek; Chandran, Aneesh; Mani, Sridhar; Dvorak, Zdenek.
Afiliação
  • Vyhlídalová B; Department of Cell Biology and Genetics, Faculty of Science, Palacky University, Slechtitelu 27, 783 71 Olomouc, Czech Republic.
  • Krasulová K; Department of Cell Biology and Genetics, Faculty of Science, Palacky University, Slechtitelu 27, 783 71 Olomouc, Czech Republic.
  • Pecinková P; Department of Cell Biology and Genetics, Faculty of Science, Palacky University, Slechtitelu 27, 783 71 Olomouc, Czech Republic.
  • Poulíková K; Department of Cell Biology and Genetics, Faculty of Science, Palacky University, Slechtitelu 27, 783 71 Olomouc, Czech Republic.
  • Vrzal R; Department of Cell Biology and Genetics, Faculty of Science, Palacky University, Slechtitelu 27, 783 71 Olomouc, Czech Republic.
  • Andrysík Z; Department of Pharmacology, University of Colorado School of Medicine, Aurora, CO 80045, USA.
  • Chandran A; Department of Medicinal Chemistry, College of Pharmacy, University of Michigan, Ann Arbor, MI 48109-1065, USA.
  • Mani S; Department of Genetics and Department of Medicine, Albert Einstein College of Medicine, Bronx, NY 10461, USA.
  • Dvorak Z; Department of Cell Biology and Genetics, Faculty of Science, Palacky University, Slechtitelu 27, 783 71 Olomouc, Czech Republic.
Int J Mol Sci ; 21(8)2020 Apr 17.
Article em En | MEDLINE | ID: mdl-32316498

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Triptaminas / Receptores de Hidrocarboneto Arílico / Citocromo P-450 CYP1A1 / Hepatócitos / Fatores de Transcrição Hélice-Alça-Hélice Básicos / Mucosa Intestinal Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Triptaminas / Receptores de Hidrocarboneto Arílico / Citocromo P-450 CYP1A1 / Hepatócitos / Fatores de Transcrição Hélice-Alça-Hélice Básicos / Mucosa Intestinal Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article