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Sirtuin 1 Inhibiting Thiocyanates (S1th)-A New Class of Isotype Selective Inhibitors of NAD+ Dependent Lysine Deacetylases.
Wössner, Nathalie; Alhalabi, Zayan; González, Jessica; Swyter, Sören; Gan, Jin; Schmidtkunz, Karin; Zhang, Lin; Vaquero, Alejandro; Ovaa, Huib; Einsle, Oliver; Sippl, Wolfgang; Jung, Manfred.
Afiliação
  • Wössner N; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg im Breisgau, Germany.
  • Alhalabi Z; Department of Medicinal Chemistry, Institute of Pharmacy, University of Halle-Wittenberg, Halle, Germany.
  • González J; Chromatin Biology Laboratory, Josep Carreras Leukaemia Research Institute (IJC), Badalona, Barcelona, Spain.
  • Swyter S; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg im Breisgau, Germany.
  • Gan J; Department of Cell and Chemical Biology, Oncode Institute, Leiden University Medical Center, Leiden, Netherlands.
  • Schmidtkunz K; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg im Breisgau, Germany.
  • Zhang L; Department of Protein Crystallography, Institute of Biochemistry, University of Freiburg, Freiburg im Breisgau, Germany.
  • Vaquero A; Chromatin Biology Laboratory, Josep Carreras Leukaemia Research Institute (IJC), Badalona, Barcelona, Spain.
  • Ovaa H; Department of Cell and Chemical Biology, Oncode Institute, Leiden University Medical Center, Leiden, Netherlands.
  • Einsle O; Department of Protein Crystallography, Institute of Biochemistry, University of Freiburg, Freiburg im Breisgau, Germany.
  • Sippl W; Department of Medicinal Chemistry, Institute of Pharmacy, University of Halle-Wittenberg, Halle, Germany.
  • Jung M; Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg im Breisgau, Germany.
Front Oncol ; 10: 657, 2020.
Article em En | MEDLINE | ID: mdl-32426286

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article