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Probing the Plasticity in the Active Site of Protein N-terminal Methyltransferase 1 Using Bisubstrate Analogues.
Chen, Dongxing; Dong, Cheng; Dong, Guangping; Srinivasan, Karthik; Min, Jinrong; Noinaj, Nicholas; Huang, Rong.
Afiliação
  • Chen D; Department of Medicinal Chemistry and Molecular Pharmacology, Center for Cancer Research, Institute for Drug Discovery, Purdue University, West Lafayette, Indiana 47907, United States.
  • Dong C; Structural Genomics Consortium, Department of Physiology, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Dong G; Department of Medicinal Chemistry and Molecular Pharmacology, Center for Cancer Research, Institute for Drug Discovery, Purdue University, West Lafayette, Indiana 47907, United States.
  • Srinivasan K; Markey Center for Structural Biology, Department of Biological Sciences and the Purdue Institute of Inflammation, Immunology and Infectious Disease, Purdue University, West Lafayette, Indiana 47907, United States.
  • Min J; Structural Genomics Consortium, Department of Physiology, University of Toronto, Toronto, Ontario M5G 1L7, Canada.
  • Noinaj N; Markey Center for Structural Biology, Department of Biological Sciences and the Purdue Institute of Inflammation, Immunology and Infectious Disease, Purdue University, West Lafayette, Indiana 47907, United States.
  • Huang R; Department of Medicinal Chemistry and Molecular Pharmacology, Center for Cancer Research, Institute for Drug Discovery, Purdue University, West Lafayette, Indiana 47907, United States.
J Med Chem ; 63(15): 8419-8431, 2020 08 13.
Article em En | MEDLINE | ID: mdl-32605369

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Domínio Catalítico / Metiltransferases Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Domínio Catalítico / Metiltransferases Limite: Humans Idioma: En Ano de publicação: 2020 Tipo de documento: Article