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Exploration of TRPM8 Binding Sites by ß-Carboline-Based Antagonists and Their In Vitro Characterization and In Vivo Analgesic Activities.
Bertamino, Alessia; Ostacolo, Carmine; Medina, Alicia; Di Sarno, Veronica; Lauro, Gianluigi; Ciaglia, Tania; Vestuto, Vincenzo; Pepe, Giacomo; Basilicata, Manuela Giovanna; Musella, Simona; Smaldone, Gerardina; Cristiano, Claudia; Gonzalez-Rodriguez, Sara; Fernandez-Carvajal, Asia; Bifulco, Giuseppe; Campiglia, Pietro; Gomez-Monterrey, Isabel; Russo, Roberto.
Afiliação
  • Bertamino A; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Ostacolo C; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
  • Medina A; IDiBE, Universitas Miguel Herna'ndez, Avda de la Universidad, 032020 Elche, Spain.
  • Di Sarno V; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Lauro G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Ciaglia T; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Vestuto V; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Pepe G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Basilicata MG; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Musella S; European Biomedical Research Institute (EBRIS), Via S. De Renzi 50, 84125 Salerno, Italy.
  • Smaldone G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Cristiano C; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
  • Gonzalez-Rodriguez S; IDiBE, Universitas Miguel Herna'ndez, Avda de la Universidad, 032020 Elche, Spain.
  • Fernandez-Carvajal A; IDiBE, Universitas Miguel Herna'ndez, Avda de la Universidad, 032020 Elche, Spain.
  • Bifulco G; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Campiglia P; Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
  • Gomez-Monterrey I; European Biomedical Research Institute (EBRIS), Via S. De Renzi 50, 84125 Salerno, Italy.
  • Russo R; Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.
J Med Chem ; 63(17): 9672-9694, 2020 09 10.
Article em En | MEDLINE | ID: mdl-32787109

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Carbolinas / Canais de Cátion TRPM / Analgésicos Limite: Animals Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Carbolinas / Canais de Cátion TRPM / Analgésicos Limite: Animals Idioma: En Ano de publicação: 2020 Tipo de documento: Article