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Synthetic group A streptogramin antibiotics that overcome Vat resistance.
Li, Qi; Pellegrino, Jenna; Lee, D John; Tran, Arthur A; Chaires, Hector A; Wang, Ruoxi; Park, Jesslyn E; Ji, Kaijie; Chow, David; Zhang, Na; Brilot, Axel F; Biel, Justin T; van Zundert, Gydo; Borrelli, Kenneth; Shinabarger, Dean; Wolfe, Cindy; Murray, Beverly; Jacobson, Matthew P; Mühle, Estelle; Chesneau, Olivier; Fraser, James S; Seiple, Ian B.
Afiliação
  • Li Q; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Pellegrino J; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, San Francisco, CA, USA.
  • Lee DJ; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, San Francisco, CA, USA.
  • Tran AA; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Chaires HA; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, San Francisco, CA, USA.
  • Wang R; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Park JE; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, San Francisco, CA, USA.
  • Ji K; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Chow D; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Zhang N; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Brilot AF; College of Life Science and Bioengineering, Beijing University of Technology, Beijing, China.
  • Biel JT; Department of Biochemistry and Biophysics and Howard Hughes Medical Institute, University of California, San Francisco, San Francisco, USA.
  • van Zundert G; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, San Francisco, CA, USA.
  • Borrelli K; Schrödinger, New York, NY, USA.
  • Shinabarger D; Department of Biochemistry and Biophysics and Howard Hughes Medical Institute, University of California, San Francisco, San Francisco, USA.
  • Wolfe C; Micromyx, Kalamazoo, MI, USA.
  • Murray B; Micromyx, Kalamazoo, MI, USA.
  • Jacobson MP; Micromyx, Kalamazoo, MI, USA.
  • Mühle E; Department of Pharmaceutical Chemistry, Cardiovascular Research Institute, University of California, San Francisco, San Francisco, CA, USA.
  • Chesneau O; Collection de l'Institut Pasteur (CIP), Microbiology Department, Institut Pasteur, Paris, France.
  • Fraser JS; Collection de l'Institut Pasteur (CIP), Microbiology Department, Institut Pasteur, Paris, France.
  • Seiple IB; Department of Bioengineering and Therapeutic Sciences, University of California, San Francisco, San Francisco, CA, USA.
Nature ; 586(7827): 145-150, 2020 10.
Article em En | MEDLINE | ID: mdl-32968273

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Estreptogramina Grupo A / Farmacorresistência Bacteriana / Antibacterianos Limite: Animals Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Estreptogramina Grupo A / Farmacorresistência Bacteriana / Antibacterianos Limite: Animals Idioma: En Ano de publicação: 2020 Tipo de documento: Article