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Addition of Fluorine and a Late-Stage Functionalization (LSF) of the Oral SERD AZD9833.
Scott, James S; Moss, Thomas A; Barlaam, Bernard; Davey, Paul R J; Fairley, Gary; Gangl, Eric T; Greenwood, Ryan D R; Hatoum-Mokdad, Holia; Lister, Andrew S; Longmire, David; Polanski, Radoslaw; Stokes, Stephen; Tucker, Michael J; Varnes, Jeffrey G; Yang, Bin.
Afiliação
  • Scott JS; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Moss TA; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Barlaam B; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Davey PRJ; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Fairley G; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Gangl ET; Oncology R&D, AstraZeneca, R&D Boston, 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Greenwood RDR; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Hatoum-Mokdad H; Oncology R&D, AstraZeneca, R&D Boston, 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Lister AS; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Longmire D; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Polanski R; Discovery Sciences, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Stokes S; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Tucker MJ; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom.
  • Varnes JG; Oncology R&D, AstraZeneca, R&D Boston, 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
  • Yang B; Oncology R&D, AstraZeneca, R&D Boston, 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.
ACS Med Chem Lett ; 11(12): 2519-2525, 2020 Dec 10.
Article em En | MEDLINE | ID: mdl-33335676

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article