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A Rationale for Drug Design Provided by Co-Crystal Structure of IC261 in Complex with Tubulin.
Xian, Jinghong; Bu, Faqian; Wang, Yuxi; Long, Fangyi; Zhang, Zhixiong; Wu, Chengyong; Tao, Yiran; Wang, Ting; Wang, Guan.
Afiliação
  • Xian J; Department of Clinical Research Management, Innovation Center of Nursing Research, Nursing Key Laboratory of Sichuan Province, West China Hospital, Collaborative Innovation Center of Biotherapy, Sichuan University, Chengdu 610041, China.
  • Bu F; Department of Clinical Research Management, Innovation Center of Nursing Research, Nursing Key Laboratory of Sichuan Province, West China Hospital, Collaborative Innovation Center of Biotherapy, Sichuan University, Chengdu 610041, China.
  • Wang Y; Precision Medicine Research Center, Department of Respiratory and Critical Care Medicine, West China Hospital, Sichuan University, Chengdu 610041, China.
  • Long F; Precision Medicine Research Center, Department of Respiratory and Critical Care Medicine, West China Hospital, Sichuan University, Chengdu 610041, China.
  • Zhang Z; Department of Pharmacy, Sichuan Cancer Hospital & Institution, Sichuan Cancer Center, School of Medicine, University of Electronic Science and Technology of China, Chengdu 610041, China.
  • Wu C; Precision Medicine Research Center, Department of Respiratory and Critical Care Medicine, West China Hospital, Sichuan University, Chengdu 610041, China.
  • Tao Y; Department of Clinical Research Management, Innovation Center of Nursing Research, Nursing Key Laboratory of Sichuan Province, West China Hospital, Collaborative Innovation Center of Biotherapy, Sichuan University, Chengdu 610041, China.
  • Wang T; Precision Medicine Research Center, Department of Respiratory and Critical Care Medicine, West China Hospital, Sichuan University, Chengdu 610041, China.
  • Wang G; Precision Medicine Research Center, Department of Respiratory and Critical Care Medicine, West China Hospital, Sichuan University, Chengdu 610041, China.
Molecules ; 26(4)2021 Feb 10.
Article em En | MEDLINE | ID: mdl-33579052

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Floroglucinol / Tubulina (Proteína) / Desenho de Fármacos / Caseína Quinase I / Indóis / Microtúbulos Limite: Animals Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Floroglucinol / Tubulina (Proteína) / Desenho de Fármacos / Caseína Quinase I / Indóis / Microtúbulos Limite: Animals Idioma: En Ano de publicação: 2021 Tipo de documento: Article