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Strained contacts with the cell membrane may influence ligand affinity to G protein coupled receptors: a case of free fatty acid receptor 1 agonists.
Lukin, Alexey; Bakholdina, Anna; Chudinov, Mikhail; Onopchenko, Oleksandra; Zhuravel, Elena; Zozulya, Sergey; Gureev, Maxim; Krasavin, Mikhail.
Afiliação
  • Lukin A; Lomonosov Institute of Fine Chemical Technologies, MIREA - Russian Technological University, Moscow, Russian Federation.
  • Bakholdina A; Lomonosov Institute of Fine Chemical Technologies, MIREA - Russian Technological University, Moscow, Russian Federation.
  • Chudinov M; Lomonosov Institute of Fine Chemical Technologies, MIREA - Russian Technological University, Moscow, Russian Federation.
  • Onopchenko O; Enamine Ltd., Kyiv, Ukraine.
  • Zhuravel E; Enamine Ltd., Kyiv, Ukraine.
  • Zozulya S; Enamine Ltd., Kyiv, Ukraine.
  • Gureev M; Taras Shevchenko National University, Kyiv, Ukraine.
  • Krasavin M; Digital Biodesign and Personalized Healthcare Research Center, Sechenov First Moscow State Medical University, Moscow, Russian Federation.
J Enzyme Inhib Med Chem ; 36(1): 1651-1658, 2021 Dec.
Article em En | MEDLINE | ID: mdl-34294008

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores Acoplados a Proteínas G / Bibliotecas de Moléculas Pequenas / Hidrazinas Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores Acoplados a Proteínas G / Bibliotecas de Moléculas Pequenas / Hidrazinas Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article