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A strategy to assess the cellular activity of E3 ligase components against neo-substrates using electrophilic probes.
Pinch, Benika J; Buckley, Dennis L; Gleim, Scott; Brittain, Scott M; Tandeske, Laura; D'Alessandro, Pier Luca; Hauseman, Zachary J; Lipps, Jennifer; Xu, Lei; Harvey, Edward P; Schirle, Markus; Sprague, Elizabeth R; Forrester, William C; Dovala, Dustin; McGregor, Lynn M; Thoma, Claudio R.
Afiliação
  • Pinch BJ; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA. Electronic address: benika.pinch@novartis.com.
  • Buckley DL; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Gleim S; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Brittain SM; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Tandeske L; Novartis Institutes for BioMedical Research, Emeryville, CA 94608, USA.
  • D'Alessandro PL; Novartis Institutes for BioMedical Research, Basel, Switzerland.
  • Hauseman ZJ; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Lipps J; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Xu L; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Harvey EP; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Schirle M; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Sprague ER; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA.
  • Forrester WC; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA. Electronic address: william.forrester@novartis.com.
  • Dovala D; Novartis Institutes for BioMedical Research, Emeryville, CA 94608, USA. Electronic address: dustin.dovala@novartis.com.
  • McGregor LM; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA. Electronic address: lynn.mcgregor@novartis.com.
  • Thoma CR; Novartis Institutes for BioMedical Research, Cambridge, MA 02139, USA. Electronic address: claudio.thoma@novartis.com.
Cell Chem Biol ; 29(1): 57-66.e6, 2022 01 20.
Article em En | MEDLINE | ID: mdl-34499862

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Ubiquitina-Proteína Ligases Limite: Female / Humans / Male Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Ubiquitina-Proteína Ligases Limite: Female / Humans / Male Idioma: En Ano de publicação: 2022 Tipo de documento: Article