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Discovery and functional characterization of N-(thiazol-2-yl)-benzamide analogs as the first class of selective antagonists of the Zinc-Activated Channel (ZAC).
Madjroh, Nawid; Mellou, Eleni; Davies, Paul A; Söderhielm, Pella C; Jensen, Anders A.
Afiliação
  • Madjroh N; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, 2100 Copenhagen Ø, Denmark.
  • Mellou E; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, 2100 Copenhagen Ø, Denmark.
  • Davies PA; Department of Neuroscience, Tufts University School of Medicine, Boston, MA, USA.
  • Söderhielm PC; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, 2100 Copenhagen Ø, Denmark.
  • Jensen AA; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, 2100 Copenhagen Ø, Denmark. Electronic address: aaj@sund.ku.dk.
Biochem Pharmacol ; 193: 114782, 2021 11.
Article em En | MEDLINE | ID: mdl-34560054

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzamidas / Receptores de Canais Iônicos de Abertura Ativada por Ligante com Alça de Cisteína / Proteínas do Tecido Nervoso Limite: Animals / Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzamidas / Receptores de Canais Iônicos de Abertura Ativada por Ligante com Alça de Cisteína / Proteínas do Tecido Nervoso Limite: Animals / Humans Idioma: En Ano de publicação: 2021 Tipo de documento: Article