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Discovery and Structure-Based Optimization of Novel Atg4B Inhibitors for the Treatment of Castration-Resistant Prostate Cancer.
Kudo, Yudai; Endo, Satoshi; Fujita, Mei; Ota, Atsumi; Kamatari, Yuji O; Tanaka, Yoshimasa; Ishikawa, Takeshi; Ikeda, Hayato; Okada, Takuya; Toyooka, Naoki; Fujimoto, Naohiro; Matsunaga, Toshiyuki; Ikari, Akira.
Afiliação
  • Kudo Y; Laboratory of Biochemistry, Gifu Pharmaceutical University, Gifu 501-1196, Japan.
  • Endo S; Laboratory of Biochemistry, Gifu Pharmaceutical University, Gifu 501-1196, Japan.
  • Fujita M; Laboratory of Biochemistry, Gifu Pharmaceutical University, Gifu 501-1196, Japan.
  • Ota A; Laboratory of Biochemistry, Gifu Pharmaceutical University, Gifu 501-1196, Japan.
  • Kamatari YO; Institute for Glyco-core Research (iGCORE), Gifu University, Gifu 501-1193, Japan.
  • Tanaka Y; United Graduate School of Drug Discovery and Medical Information Sciences, Gifu University, Gifu 501-1193, Japan.
  • Ishikawa T; Center for Medical Innovation, Nagasaki University, 1-7-1 Sakamoto, Nagasaki 852-8588, Japan.
  • Ikeda H; Graduate School of Science and Engineering, Kagoshima University, 1-21-40 Korimoto, Kagoshima 890-0065, Japan.
  • Okada T; Graduate School of Innovative Life Science, University of Toyama, Toyama 930-8555, Japan.
  • Toyooka N; Graduate School of Innovative Life Science, University of Toyama, Toyama 930-8555, Japan.
  • Fujimoto N; Graduate School of Innovative Life Science, University of Toyama, Toyama 930-8555, Japan.
  • Matsunaga T; Department of Urology, University of Occupational and Environmental Health, Kitakyushu 807-8555, Japan.
  • Ikari A; Education Center of Green Pharmaceutical Sciences, Gifu Pharmaceutical University, Gifu 502-8585, Japan.
J Med Chem ; 65(6): 4878-4892, 2022 03 24.
Article em En | MEDLINE | ID: mdl-35244402

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias de Próstata Resistentes à Castração Tipo de estudo: Prognostic_studies Limite: Humans / Male Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias de Próstata Resistentes à Castração Tipo de estudo: Prognostic_studies Limite: Humans / Male Idioma: En Ano de publicação: 2022 Tipo de documento: Article