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Overcoming Paradoxical Kinase Priming by a Novel MNK1 Inhibitor.
Bou-Petit, Elisabeth; Hümmer, Stefan; Alarcon, Helena; Slobodnyuk, Konstantin; Cano-Galietero, Marta; Fuentes, Pedro; Guijarro, Pedro J; Muñoz, María José; Suarez-Cabrera, Leticia; Santamaria, Anna; Estrada-Tejedor, Roger; Borrell, José I; Ramón Y Cajal, Santiago.
Afiliação
  • Bou-Petit E; Grup de Química Farmacèutica, IQS School of Engineering, Universitat Ramon Llull, Via Augusta, 390, 08017 Barcelona, Spain.
  • Hümmer S; Translational Molecular Pathology, Vall d'Hebron Research Institute (VHIR), Universitat Autònoma de Barcelona, Psg. Vall d'Hebron 119-129, 08035 Barcelona, Spain.
  • Alarcon H; Spanish Biomedical Research Network Centre in Oncology (CIBERONC), 28029 Madrid, Spain.
  • Slobodnyuk K; Grup de Química Farmacèutica, IQS School of Engineering, Universitat Ramon Llull, Via Augusta, 390, 08017 Barcelona, Spain.
  • Cano-Galietero M; Translational Molecular Pathology, Vall d'Hebron Research Institute (VHIR), Universitat Autònoma de Barcelona, Psg. Vall d'Hebron 119-129, 08035 Barcelona, Spain.
  • Fuentes P; Spanish Biomedical Research Network Centre in Oncology (CIBERONC), 28029 Madrid, Spain.
  • Guijarro PJ; Translational Molecular Pathology, Vall d'Hebron Research Institute (VHIR), Universitat Autònoma de Barcelona, Psg. Vall d'Hebron 119-129, 08035 Barcelona, Spain.
  • Muñoz MJ; Spanish Biomedical Research Network Centre in Oncology (CIBERONC), 28029 Madrid, Spain.
  • Suarez-Cabrera L; Translational Molecular Pathology, Vall d'Hebron Research Institute (VHIR), Universitat Autònoma de Barcelona, Psg. Vall d'Hebron 119-129, 08035 Barcelona, Spain.
  • Santamaria A; Spanish Biomedical Research Network Centre in Oncology (CIBERONC), 28029 Madrid, Spain.
  • Estrada-Tejedor R; Translational Molecular Pathology, Vall d'Hebron Research Institute (VHIR), Universitat Autònoma de Barcelona, Psg. Vall d'Hebron 119-129, 08035 Barcelona, Spain.
  • Borrell JI; Translational Molecular Pathology, Vall d'Hebron Research Institute (VHIR), Universitat Autònoma de Barcelona, Psg. Vall d'Hebron 119-129, 08035 Barcelona, Spain.
  • Ramón Y Cajal S; Spanish Biomedical Research Network Centre in Oncology (CIBERONC), 28029 Madrid, Spain.
J Med Chem ; 65(8): 6070-6087, 2022 04 28.
Article em En | MEDLINE | ID: mdl-35417652

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas Serina-Treonina Quinases / Peptídeos e Proteínas de Sinalização Intracelular Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas Serina-Treonina Quinases / Peptídeos e Proteínas de Sinalização Intracelular Idioma: En Ano de publicação: 2022 Tipo de documento: Article