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Identification of parallel medicinal chemistry protocols to expand branched amine design space.
Conn, Edward L; Perry, Matthew A; Shi, Kecheng; Wang, Guotao; Hoy, Susan; Sach, Neal W; Qi, Wenying; Qu, Liqiang; Gao, Yu; Xu, Yan; Schmitt, Daniel C.
Afiliação
  • Conn EL; Medicine Design, Pfizer Worldwide Research, Development and Medical, Groton, Connecticut 06340, USA. daniel.schmitt@pfizer.com.
  • Perry MA; Medicine Design, Pfizer Worldwide Research, Development and Medical, Groton, Connecticut 06340, USA. daniel.schmitt@pfizer.com.
  • Shi K; WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.
  • Wang G; WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.
  • Hoy S; Medicine Design, Pfizer Worldwide Research, Development and Medical, Groton, Connecticut 06340, USA. daniel.schmitt@pfizer.com.
  • Sach NW; Medicine Design, Pfizer Worldwide Research, Development and Medical, 10770 Science Center Drive, San Diego, California 92121, USA.
  • Qi W; WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.
  • Qu L; WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.
  • Gao Y; WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.
  • Xu Y; WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China.
  • Schmitt DC; Medicine Design, Pfizer Worldwide Research, Development and Medical, Groton, Connecticut 06340, USA. daniel.schmitt@pfizer.com.
Org Biomol Chem ; 20(18): 3747-3754, 2022 05 11.
Article em En | MEDLINE | ID: mdl-35448901

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Química Farmacêutica / Aminas Tipo de estudo: Diagnostic_studies Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Química Farmacêutica / Aminas Tipo de estudo: Diagnostic_studies Idioma: En Ano de publicação: 2022 Tipo de documento: Article