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Interaction of letrozole and its degradation products with aromatase: chemometric assessment of kinetics and structure-based binding validation.
De Luca, Michele; Occhiuzzi, Maria Antonietta; Rizzuti, Bruno; Ioele, Giuseppina; Ragno, Gaetano; Garofalo, Antonio; Grande, Fedora.
Afiliação
  • De Luca M; Department of Pharmacy, Health and Nutritional Sciences, University of Calabria, Rende, Italy.
  • Occhiuzzi MA; Department of Pharmacy, Health and Nutritional Sciences, University of Calabria, Rende, Italy.
  • Rizzuti B; CNR-NANOTEC, SS Rende (CS), Department of Physics, University of Calabria, Rende, Italy.
  • Ioele G; Institute for Biocomputation and Physics of Complex Systems (BIFI), Joint Unit GBsC-CSIC-BIFI, University of Zaragoza, Zaragoza, Spain.
  • Ragno G; Department of Pharmacy, Health and Nutritional Sciences, University of Calabria, Rende, Italy.
  • Garofalo A; Department of Pharmacy, Health and Nutritional Sciences, University of Calabria, Rende, Italy.
  • Grande F; Department of Pharmacy, Health and Nutritional Sciences, University of Calabria, Rende, Italy.
J Enzyme Inhib Med Chem ; 37(1): 1600-1609, 2022 Dec.
Article em En | MEDLINE | ID: mdl-35635194

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Aromatase / Inibidores da Aromatase Limite: Female / Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Aromatase / Inibidores da Aromatase Limite: Female / Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article