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Stereoselective synthesis of 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as PIM kinase inhibitors inspired from marine alkaloids.
Casuscelli, Francesco; Ardini, Elena; Avanzi, Nilla; Badari, Alessandra; Casale, Elena; Disingrini, Teresa; Donati, Daniele; Ermoli, Antonella; Felder, Eduard R; Galvani, Arturo; Isacchi, Antonella; Menichincheri, Maria; Montemartini, Marisa; Orrenius, Christian; Piutti, Claudia; Salom, Barbara; Papeo, Gianluca.
Afiliação
  • Casuscelli F; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Ardini E; Accelera, Nerviano Medical Sciences, Nerviano, Milan, Italy.
  • Avanzi N; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Badari A; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Casale E; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Disingrini T; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Donati D; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Ermoli A; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Felder ER; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Galvani A; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Isacchi A; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Menichincheri M; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Montemartini M; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Orrenius C; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Piutti C; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
  • Salom B; Accelera, Nerviano Medical Sciences, Nerviano, Milan, Italy.
  • Papeo G; Oncology, Nerviano Medical Sciences, Nerviano (Mi), Italy.
Chirality ; 34(11): 1437-1452, 2022 11.
Article em En | MEDLINE | ID: mdl-35959859

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Alcaloides / Antineoplásicos Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Alcaloides / Antineoplásicos Idioma: En Ano de publicação: 2022 Tipo de documento: Article