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Enantioselective Approach for Expanding the Three-Dimensional Space of Tetrahydroquinoline to Develop BET Bromodomain Inhibitors.
Lespinasse, Marie-Ange; Wei, Kaiyao; Perrin, Justine; Winkler, Matthias; Hamaidia, Sieme; Leroy, Alexis; Macek Jilkova, Zuzana; Philouze, Christian; Marche, Patrice N; Petosa, Carlo; Govin, Jérôme; Emadali, Anouk; Wong, Yung-Sing.
Afiliação
  • Lespinasse MA; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France.
  • Wei K; Univ. Grenoble Alpes, Inserm U1209, CNRS 5309, IAB, 38000, Grenoble, France.
  • Perrin J; Univ. Grenoble Alpes, CEA, CNRS 5075, IBS, 38000, Grenoble, France.
  • Winkler M; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France.
  • Hamaidia S; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France.
  • Leroy A; Univ. Grenoble Alpes, Inserm U1209, CNRS 5309, IAB, 38000, Grenoble, France.
  • Macek Jilkova Z; Univ. Grenoble Alpes, Inserm U1209, CNRS 5309, IAB, 38000, Grenoble, France.
  • Philouze C; Univ. Grenoble Alpes, Inserm U1209, CNRS 5309, IAB, 38000, Grenoble, France.
  • Marche PN; Univ. Grenoble Alpes, CHU Grenoble Alpes, 38000, Grenoble, France.
  • Petosa C; Univ. Grenoble Alpes, CNRS 5250, DCM, 38000, Grenoble, France.
  • Govin J; Univ. Grenoble Alpes, Inserm U1209, CNRS 5309, IAB, 38000, Grenoble, France.
  • Emadali A; Univ. Grenoble Alpes, CEA, CNRS 5075, IBS, 38000, Grenoble, France.
  • Wong YS; Univ. Grenoble Alpes, Inserm U1209, CNRS 5309, IAB, 38000, Grenoble, France.
Chemistry ; 28(64): e202202293, 2022 Nov 16.
Article em En | MEDLINE | ID: mdl-35989226

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Antineoplásicos Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Antineoplásicos Idioma: En Ano de publicação: 2022 Tipo de documento: Article