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Revisiting a challenging p53 binding site: a diversity-optimized HEFLib reveals diverse binding modes in T-p53C-Y220C.
Stahlecker, Jason; Klett, Theresa; Schwer, Martin; Jaag, Simon; Dammann, Marcel; Ernst, Larissa N; Braun, Michael B; Zimmermann, Markus O; Kramer, Markus; Lämmerhofer, Michael; Stehle, Thilo; Coles, Murray; Boeckler, Frank M.
Afiliação
  • Stahlecker J; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
  • Klett T; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
  • Schwer M; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
  • Jaag S; Institute of Pharmaceutical Sciences, Pharmaceutical (Bio-)Analysis, University of Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany.
  • Dammann M; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
  • Ernst LN; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
  • Braun MB; Interfaculty Institute of Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 34 72076 Tübingen Germany.
  • Zimmermann MO; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
  • Kramer M; Institute of Organic Chemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 18 72076 Tübingen Germany.
  • Lämmerhofer M; Institute of Pharmaceutical Sciences, Pharmaceutical (Bio-)Analysis, University of Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany.
  • Stehle T; Interfaculty Institute of Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 34 72076 Tübingen Germany.
  • Coles M; Department of Protein Evolution, Max Planck Institute for Biology Tübingen Max-Planck-Ring 5 72076 Tübingen Germany.
  • Boeckler FM; Lab for Molecular Design & Pharm. Biophysics, Institute of Pharmaceutical Sciences, Department of Pharmacy and Biochemistry, Eberhard Karls Universität Tübingen Auf der Morgenstelle 8 72076 Tübingen Germany frank.boeckler@uni-tuebingen.de.
RSC Med Chem ; 13(12): 1575-1586, 2022 Dec 14.
Article em En | MEDLINE | ID: mdl-36561072

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Ano de publicação: 2022 Tipo de documento: Article