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Design, Synthesis, and Pharmacological Evaluation of Embelin-Aryl/alkyl Amine Hybrids as Orally Bioavailable Blood-Brain Barrier Permeable Multitargeted Agents with Therapeutic Potential in Alzheimer's Disease: Discovery of SB-1448.
Nuthakki, Vijay K; Choudhary, Sushil; Reddy, Chilakala N; Bhatt, Shipra; Jamwal, Ashiya; Jotshi, Anshika; Raghuvanshi, Rinky; Sharma, Ankita; Thakur, Shikha; Jadhav, Hemant R; Bharate, Sonali S; Nandi, Utpal; Kumar, Ajay; Bharate, Sandip B.
Afiliação
  • Nuthakki VK; Natural Products & Medicinal Chemistry Division, CSIR-Indian Institute of Integrative Medicine, Canal Road, Jammu 180001, India.
  • Choudhary S; Academy of Scientific & Innovative Research (AcSIR), Ghaziabad 201002, India.
  • Reddy CN; Pharmacology Division, CSIR-Indian Institute of Integrative Medicine, Jammu 180001, India.
  • Bhatt S; Academy of Scientific & Innovative Research (AcSIR), Ghaziabad 201002, India.
  • Jamwal A; Natural Products & Medicinal Chemistry Division, CSIR-Indian Institute of Integrative Medicine, Canal Road, Jammu 180001, India.
  • Jotshi A; Academy of Scientific & Innovative Research (AcSIR), Ghaziabad 201002, India.
  • Raghuvanshi R; Pharmacology Division, CSIR-Indian Institute of Integrative Medicine, Jammu 180001, India.
  • Sharma A; Academy of Scientific & Innovative Research (AcSIR), Ghaziabad 201002, India.
  • Thakur S; Pharmacology Division, CSIR-Indian Institute of Integrative Medicine, Jammu 180001, India.
  • Jadhav HR; Academy of Scientific & Innovative Research (AcSIR), Ghaziabad 201002, India.
  • Bharate SS; Pharmacology Division, CSIR-Indian Institute of Integrative Medicine, Jammu 180001, India.
  • Nandi U; Natural Products & Medicinal Chemistry Division, CSIR-Indian Institute of Integrative Medicine, Canal Road, Jammu 180001, India.
  • Kumar A; Academy of Scientific & Innovative Research (AcSIR), Ghaziabad 201002, India.
  • Bharate SB; Natural Products & Medicinal Chemistry Division, CSIR-Indian Institute of Integrative Medicine, Canal Road, Jammu 180001, India.
ACS Chem Neurosci ; 14(6): 1193-1219, 2023 03 15.
Article em En | MEDLINE | ID: mdl-36812360

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Doença de Alzheimer Tipo de estudo: Risk_factors_studies Limite: Animals / Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Doença de Alzheimer Tipo de estudo: Risk_factors_studies Limite: Animals / Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article