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Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9.
Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi.
Afiliação
  • Gazzillo E; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy; PhD Program in Drug Discovery and Development, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy.
  • Pierri M; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy; PhD Program in Drug Discovery and Development, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy.
  • Colarusso E; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy.
  • Chini MG; Department of Biosciences and Territory, University of Molise, C.da Fonte Lappone, Pesche 86090, Italy.
  • Ferraro MG; BioChem Lab, Department of Pharmacy, School of Medicine and Surgery, University of Naples, Via Domenico Montesano 49, Naples 80131, Italy.
  • Piccolo M; BioChem Lab, Department of Pharmacy, School of Medicine and Surgery, University of Naples, Via Domenico Montesano 49, Naples 80131, Italy.
  • Irace C; BioChem Lab, Department of Pharmacy, School of Medicine and Surgery, University of Naples, Via Domenico Montesano 49, Naples 80131, Italy.
  • Bruno I; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy.
  • Bifulco G; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy.
  • Terracciano S; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy. Electronic address: sterracciano@unisa.it.
  • Lauro G; Department of Pharmacy, University of Salerno, Via Giovanni Paolo II 132, Fisciano 84084, Italy. Electronic address: glauro@unisa.it.
Bioorg Chem ; 139: 106677, 2023 10.
Article em En | MEDLINE | ID: mdl-37352721

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Leucemia Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Leucemia Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article