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Structural Fusion of Natural and Synthetic Ligand Features Boosts RXR Agonist Potency.
Adouvi, Gustave; Nawa, Felix; Ballarotto, Marco; Rüger, Lorena Andrea; Knümann, Loris; Kasch, Till; Arifi, Silvia; Schubert-Zsilavecz, Manfred; Willems, Sabine; Marschner, Julian A; Pabel, Jörg; Merk, Daniel.
Afiliação
  • Adouvi G; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Nawa F; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Ballarotto M; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Rüger LA; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Knümann L; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Kasch T; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Arifi S; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Schubert-Zsilavecz M; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Willems S; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Marschner JA; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Pabel J; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Merk D; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
J Med Chem ; 66(24): 16762-16771, 2023 12 28.
Article em En | MEDLINE | ID: mdl-38064686

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Acrilatos / Receptores do Ácido Retinoico Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Acrilatos / Receptores do Ácido Retinoico Idioma: En Ano de publicação: 2023 Tipo de documento: Article