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In silico Design, Synthesis and Biological Evaluation of Novel Thieno[3,2-d]pyrimidine Derivatives for Cancer Therapy - A Preliminary Study on the Inhibitory Potential towards ATR Kinase Domain and PIKK Family.
Sirakanyan, Samvel N; Dilip, Haritha; Geronikaki, Athina; Spinelli, Domenico; Kirubakaran, Sivapriya; Petrou, Anthi; Hakobyan, Elmira K; Kartsev, Victor G; Paronikyan, Ervand G; Yegoryan, Hasmik A; Yermalovyan, Lilit V; Hovakimyan, Anush A.
Afiliação
  • Sirakanyan SN; Scientific Technological Center of Organic and Pharmaceutical Chemistry of National Academy of Science of Republic of Armenia, Institute of Fine Organic Chemistry of A.L.Mnjoyan, Ave., Azatutyan 26, Yerevan, 0014, Armenia.
  • Dilip H; Department of Chemistry, Indian Institute of Technology Gandhinagar, Palaj Village, Gandhinagar, Gujarat, 382055, India.
  • Geronikaki A; School of Pharmacy, Aristotle University of Thessaloniki, 54124, Thessaloniki, Greece.
  • Spinelli D; Dipartimento di Chimica G. Ciamician, Alma Mater Studiorum-Università di Bologna, Via F. Selmi 2, 40126, Bologna, Italy.
  • Kirubakaran S; Department of Chemistry, Indian Institute of Technology Gandhinagar, Palaj Village, Gandhinagar, Gujarat, 382055, India.
  • Petrou A; School of Pharmacy, Aristotle University of Thessaloniki, 54124, Thessaloniki, Greece.
  • Hakobyan EK; Scientific Technological Center of Organic and Pharmaceutical Chemistry of National Academy of Science of Republic of Armenia, Institute of Fine Organic Chemistry of A.L.Mnjoyan, Ave., Azatutyan 26, Yerevan, 0014, Armenia.
  • Kartsev VG; InterBioScreen, Moscow, 119019, Russia.
  • Paronikyan EG; Scientific Technological Center of Organic and Pharmaceutical Chemistry of National Academy of Science of Republic of Armenia, Institute of Fine Organic Chemistry of A.L.Mnjoyan, Ave., Azatutyan 26, Yerevan, 0014, Armenia.
  • Yegoryan HA; Scientific Technological Center of Organic and Pharmaceutical Chemistry of National Academy of Science of Republic of Armenia, Institute of Fine Organic Chemistry of A.L.Mnjoyan, Ave., Azatutyan 26, Yerevan, 0014, Armenia.
  • Yermalovyan LV; Scientific Technological Center of Organic and Pharmaceutical Chemistry of National Academy of Science of Republic of Armenia, Institute of Fine Organic Chemistry of A.L.Mnjoyan, Ave., Azatutyan 26, Yerevan, 0014, Armenia.
  • Hovakimyan AA; Scientific Technological Center of Organic and Pharmaceutical Chemistry of National Academy of Science of Republic of Armenia, Institute of Fine Organic Chemistry of A.L.Mnjoyan, Ave., Azatutyan 26, Yerevan, 0014, Armenia.
Chem Biodivers ; 21(3): e202302071, 2024 Mar.
Article em En | MEDLINE | ID: mdl-38230843

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias / Antineoplásicos Idioma: En Ano de publicação: 2024 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Neoplasias / Antineoplásicos Idioma: En Ano de publicação: 2024 Tipo de documento: Article