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Synthesis and in vitro evaluation of diverse heterocyclic diphenolic compounds as inhibitors of DYRK1A.
Zhou, Qingqing; Reekie, Tristan A; Abbassi, Ramzi H; Indurthi Venkata, Dinesh; Font, Josep S; Ryan, Renae M; Munoz, Lenka; Kassiou, Michael.
Afiliação
  • Zhou Q; School of Chemistry, The University of Sydney, New South Wales 2006, Australia.
  • Reekie TA; School of Chemistry, The University of Sydney, New South Wales 2006, Australia.
  • Abbassi RH; School of Medical Sciences, Discipline of Pathology and Charles Perkins Centre, The University of Sydney, New South Wales 2006, Australia.
  • Indurthi Venkata D; School of Medical Sciences, Discipline of Pathology and Charles Perkins Centre, The University of Sydney, New South Wales 2006, Australia.
  • Font JS; School of Medical Sciences, Discipline of Pharmacology, The University of Sydney, New South Wales 2006, Australia.
  • Ryan RM; School of Medical Sciences, Discipline of Pharmacology, The University of Sydney, New South Wales 2006, Australia.
  • Munoz L; School of Medical Sciences, Discipline of Pathology and Charles Perkins Centre, The University of Sydney, New South Wales 2006, Australia.
  • Kassiou M; School of Chemistry, The University of Sydney, New South Wales 2006, Australia. Electronic address: michael.kassiou@sydney.edu.au.
Bioorg Med Chem ; 26(22): 5852-5869, 2018 12 01.
Article em En | MEDLINE | ID: mdl-30401502

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fenóis / Proteínas Tirosina Quinases / Proteínas Serina-Treonina Quinases / Inibidores de Proteínas Quinases / Compostos Heterocíclicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Austrália País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fenóis / Proteínas Tirosina Quinases / Proteínas Serina-Treonina Quinases / Inibidores de Proteínas Quinases / Compostos Heterocíclicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Austrália País de publicação: Reino Unido