1.
Bioorg Med Chem Lett
; 14(11): 2955-8, 2004 Jun 07.
Article
in English
| MEDLINE
| ID: mdl-15125967
ABSTRACT
A series of purine based inhibitors of PDE7 has been derived from screening lead 1a. The synthesis, structure-activity relationships (SAR), and selectivity against several other PDE family members are described.