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1.
Modulation of macrophage inflammatory function through selective inhibition of the epigenetic reader protein SP140.
BMC Biol
; 20(1): 182, 2022 08 19.
Article
in English
| MEDLINE | ID: mdl-35986286
2.
Preclinical candidate for the treatment of visceral leishmaniasis that acts through proteasome inhibition.
Proc Natl Acad Sci U S A
; 116(19): 9318-9323, 2019 05 07.
Article
in English
| MEDLINE | ID: mdl-30962368
3.
Structure guided drug design to develop kallikrein 5 inhibitors to treat Netherton syndrome.
Bioorg Med Chem Lett
; 29(12): 1454-1458, 2019 06 15.
Article
in English
| MEDLINE | ID: mdl-31005442
4.
Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors.
Bioorg Med Chem Lett
; 29(20): 126675, 2019 10 15.
Article
in English
| MEDLINE | ID: mdl-31521475
5.
Inhibition of PAD4 activity is sufficient to disrupt mouse and human NET formation.
Nat Chem Biol
; 11(3): 189-91, 2015 Mar.
Article
in English
| MEDLINE | ID: mdl-25622091
6.
Corrigendum to 'Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors' [Bioorg. Med. Chem. Lett. 29 (2019) 126675].
Bioorg Med Chem Lett
; 30(2): 126771, 2020 Jan 15.
Article
in English
| MEDLINE | ID: mdl-31859161
7.
Reducing False Positives through the Application of Fluorescence Lifetime Technology: A Comparative Study Using TYK2 Kinase as a Model System.
SLAS Discov
; 26(5): 663-675, 2021 06.
Article
in English
| MEDLINE | ID: mdl-33783261
8.
Novel Selection Approaches to Identify Antibodies Targeting Neoepitopes on the C5b6 Intermediate Complex to Inhibit Membrane Attack Complex Formation.
Antibodies (Basel)
; 10(4)2021 Oct 12.
Article
in English
| MEDLINE | ID: mdl-34698051
9.
Structurally Diverse Mitochondrial Branched Chain Aminotransferase (BCATm) Leads with Varying Binding Modes Identified by Fragment Screening.
J Med Chem
; 59(6): 2452-67, 2016 Mar 24.
Article
in English
| MEDLINE | ID: mdl-26938474
10.
The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits.
J Med Chem
; 58(18): 7140-63, 2015 Sep 24.
Article
in English
| MEDLINE | ID: mdl-26090771
11.
A modular, fully integrated ultra-high-throughput screening system based on confocal fluorescence analysis techniques.
J Biomol Screen
; 8(6): 648-59, 2003 Dec.
Article
in English
| MEDLINE | ID: mdl-14711390
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