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1.
Discovery of low-molecular-weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability.
J Med Virol
; 96(4): e29594, 2024 Apr.
Article
in English
| MEDLINE | ID: mdl-38576317
2.
Discovery of novel 1,2,4-triazole phenylalanine derivatives targeting an unexplored region within the interprotomer pocket of the HIV capsid protein.
J Med Virol
; 94(12): 5975-5986, 2022 12.
Article
in English
| MEDLINE | ID: mdl-35949003
3.
Discovery of Novel Boron-Containing N-Substituted Oseltamivir Derivatives as Anti-Influenza A Virus Agents for Overcoming N1-H274Y Oseltamivir-Resistant.
Molecules
; 27(19)2022 Sep 29.
Article
in English
| MEDLINE | ID: mdl-36234966
4.
Design, Synthesis, and Evaluation of a Set of Carboxylic Acid and Phosphate Prodrugs Derived from HBV Capsid Protein Allosteric Modulator NVR 3-778.
Molecules
; 27(18)2022 Sep 14.
Article
in English
| MEDLINE | ID: mdl-36144715
5.
Design, Synthesis and Structure-Activity Relationships of Phenylalanine-Containing Peptidomimetics as Novel HIV-1 Capsid Binders Based on Ugi Four-Component Reaction.
Molecules
; 27(18)2022 Sep 14.
Article
in English
| MEDLINE | ID: mdl-36144727
6.
Design, synthesis, and antiviral activity of phenylalanine derivatives as HIV-1 capsid inhibitors.
Bioorg Med Chem
; 48: 116414, 2021 10 15.
Article
in English
| MEDLINE | ID: mdl-34562701
7.
Discovery of novel diarypyrimidine derivatives bearing six-membered non-aromatic heterocycles as potent HIV-1 NNRTIs with improved anti-resistance and drug-like profiles.
Eur J Med Chem
; 258: 115605, 2023 Oct 05.
Article
in English
| MEDLINE | ID: mdl-37393790
8.
Discovery of diarylpyrimidine derivatives bearing piperazine sulfonyl as potent HIV-1 nonnucleoside reverse transcriptase inhibitors.
Commun Chem
; 6(1): 83, 2023 Apr 29.
Article
in English
| MEDLINE | ID: mdl-37120482
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