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1.
Electrochemical Synthesis of 2-Aryl-3-(2-aminoaryl)quinoxalines via Oxidative Dearomatization/Ring-Opening/Cyclization Cascade Sequence of 2-Arylindoles with 1,2-Diaminoarenes.
J Org Chem
; 88(15): 11111-11121, 2023 Aug 04.
Article
in English
| MEDLINE | ID: mdl-37489614
2.
Electrochemical Oxidative Addition of Nucleophiles on 2-Arylindoles: Synthesis of C2-Heteroquaternary Indolin-3-ones.
J Org Chem
; 87(23): 15771-15782, 2022 Dec 02.
Article
in English
| MEDLINE | ID: mdl-36394546
3.
Design, synthesis and biological evaluation studies of novel small molecule ENPP1 inhibitors for cancer immunotherapy.
Bioorg Chem
; 119: 105549, 2022 02.
Article
in English
| MEDLINE | ID: mdl-34929517
4.
Electrochemical Oxidative Coupling Between Benzylic C(sp3)-H and N-H of Secondary Amines: Rapid Synthesis of α-Amino α-Aryl Esters.
J Org Chem
; 86(14): 9682-9691, 2021 07 16.
Article
in English
| MEDLINE | ID: mdl-34184902
5.
Identification and structure-activity relationship studies of small molecule inhibitors of the human cathepsin D.
Bioorg Med Chem
; 29: 115879, 2021 01 01.
Article
in English
| MEDLINE | ID: mdl-33271453
6.
Direct Amine-Catalyzed Enantioselective Synthesis of Pentacyclic Dibenzo[b,f][1,4]oxazepine/Thiazepine-Fused Isoquinuclidines along with DFT Calculations.
J Org Chem
; 85(21): 14094-14108, 2020 11 06.
Article
in English
| MEDLINE | ID: mdl-33030896
7.
Enantioselective Direct Synthesis of C3-Hydroxyalkylated Pyrrole via an Amine-Catalyzed Aldol/Paal-Knorr Reaction Sequence.
Org Lett
; 24(41): 7549-7554, 2022 Oct 21.
Article
in English
| MEDLINE | ID: mdl-36219141
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