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1.
Inhibition of Prolyl Oligopeptidase Restores Prohibitin 2 Levels in Psychosis Models: Relationship to Cognitive Deficits in Schizophrenia.
Int J Mol Sci
; 24(7)2023 Mar 23.
Article
in English
| MEDLINE | ID: mdl-37046989
2.
Design and synthesis of selective and blood-brain barrier-permeable hydroxamate-based gelatinase inhibitors.
Bioorg Chem
; 94: 103365, 2020 01.
Article
in English
| MEDLINE | ID: mdl-31676116
3.
Applying the retro-enantio approach to obtain a peptide capable of overcoming the blood-brain barrier.
Angew Chem Int Ed Engl
; 54(13): 3967-72, 2015 Mar 23.
Article
in English
| MEDLINE | ID: mdl-25650865
4.
Dual system for the central nervous system targeting and blood-brain barrier transport of a selective prolyl oligopeptidase inhibitor.
Biopolymers
; 100(6): 662-74, 2013 Nov.
Article
in English
| MEDLINE | ID: mdl-23893478
5.
Peptidomimetics designed to bind to RAS effector domain are promising cancer therapeutic compounds.
Sci Rep
; 12(1): 15810, 2022 09 22.
Article
in English
| MEDLINE | ID: mdl-36138080
6.
The Gelatinase Inhibitor ACT-03 Reduces Gliosis in the Rapid Kindling Rat Model of Epilepsy, and Attenuates Inflammation and Loss of Barrier Integrity In Vitro.
Biomedicines
; 10(9)2022 Aug 29.
Article
in English
| MEDLINE | ID: mdl-36140216
7.
Rational design of a selective covalent modifier of G protein ßγ subunits.
Mol Pharmacol
; 79(1): 24-33, 2011 Jan.
Article
in English
| MEDLINE | ID: mdl-20881007
8.
The matrix metalloproteinase inhibitor IPR-179 has antiseizure and antiepileptogenic effects.
J Clin Invest
; 131(1)2021 01 04.
Article
in English
| MEDLINE | ID: mdl-33141761
9.
A MALDI-TOF-based Method for Studying the Transport of BBB Shuttles-Enhancing Sensitivity and Versatility of Cell-Based In Vitro Transport Models.
Sci Rep
; 9(1): 4875, 2019 03 19.
Article
in English
| MEDLINE | ID: mdl-30890722
10.
Molecular basis for the protective effects of low-density lipoprotein receptor-related protein 1 (LRP1)-derived peptides against LDL aggregation.
Biochim Biophys Acta Biomembr
; 1861(7): 1302-1316, 2019 07 01.
Article
in English
| MEDLINE | ID: mdl-31077676
11.
Baicalin, a prodrug able to reach the CNS, is a prolyl oligopeptidase inhibitor.
Bioorg Med Chem
; 16(15): 7516-24, 2008 Aug 01.
Article
in English
| MEDLINE | ID: mdl-18650094
12.
HAI Peptide and Backbone Analogs-Validation and Enhancement of Biostability and Bioactivity of BBB Shuttles.
Sci Rep
; 8(1): 17932, 2018 12 18.
Article
in English
| MEDLINE | ID: mdl-30560894
13.
Targeted Covalent Inhibition of Prolyl Oligopeptidase (POP): Discovery of Sulfonylfluoride Peptidomimetics.
Cell Chem Biol
; 25(8): 1031-1037.e4, 2018 08 16.
Article
in English
| MEDLINE | ID: mdl-29779956
14.
The prolyl oligopeptidase inhibitor IPR19 ameliorates cognitive deficits in mouse models of schizophrenia.
Eur Neuropsychopharmacol
; 27(2): 180-191, 2017 02.
Article
in English
| MEDLINE | ID: mdl-27986355
15.
The glial phosphorylase of glycogen isoform is reduced in the dorsolateral prefrontal cortex in chronic schizophrenia.
Schizophr Res
; 177(1-3): 37-43, 2016 11.
Article
in English
| MEDLINE | ID: mdl-27156240
16.
A novel family of diketopiperazines as a tool for the study of transport across the blood-brain barrier (BBB) and their potential use as BBB-shuttles.
Adv Exp Med Biol
; 611: 227-8, 2009.
Article
in English
| MEDLINE | ID: mdl-19400172
17.
Increased SP4 and SP1 transcription factor expression in the postmortem hippocampus of chronic schizophrenia.
J Psychiatr Res
; 58: 189-96, 2014 Nov.
Article
in English
| MEDLINE | ID: mdl-25175639
18.
Peptide POP inhibitors for the treatment of the cognitive symptoms of schizophrenia.
Future Med Chem
; 5(13): 1509-23, 2013 Sep.
Article
in English
| MEDLINE | ID: mdl-24024944
19.
Delivery of gold nanoparticles to the brain by conjugation with a peptide that recognizes the transferrin receptor.
Biomaterials
; 33(29): 7194-205, 2012 Oct.
Article
in English
| MEDLINE | ID: mdl-22795856
20.
N-methyl phenylalanine-rich peptides as highly versatile blood-brain barrier shuttles.
J Med Chem
; 53(6): 2354-63, 2010 Mar 25.
Article
in English
| MEDLINE | ID: mdl-20170117
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